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ARYL AND HETEROARYL MORPHOLINE DERIVATIVES

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专利名称:ARYL AND HETEROARYL MORPHOLINE

DERIVATIVES

发明人:CASES-THOMAS, Manuel, Javier,HAUGHTON,

Helen, Louise,LAMAS-PETEIRA,Carlos,OUWERKERK-MAHADEVAN,Sivi,MASTERS, John, Joseph,SIMMONDS,Robin, George,RUDYK, Hélène, Catherine,Eugénie,WALTER, Magnus, Wilhelm

申请号:EP037475.4申请日:20030818公开号:EP1534694A1公开日:20050601

摘要:Compounds of formula (I) are selective inhibitors of the reuptake of

norepinephrine, wherein Rx is H; Ry is H or C1-C4 alkyl; each Rz is independently H or C1-C4 alkyl; X represents O; Y represents OH or OR; R is C1-C4 alkyl; and Ar1 and Ar2 areoptionally substituted phenyl or 5- or 6-membered heteroaryl rings.

申请人:ELI LILLY AND COMPANY

地址:Lilly Corporate Center Indianapolis, Indiana 46285 US

国籍:US

代理机构:Kingsbury, Oliver William

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